Recent advance in direct sp3 carbon‐hydrogen bond functionalizations
نویسندگان
چکیده
Received: 20 February 2016 Accepted: 19 March 2016 Published online: 30 June 2016 Printed: 30 June 2016 Direct and selective carbon‐hydrogen bond functionalization has attracted enormous attention because it provides more efficient strategies for preparing valuable functional molecules from easily available substrates. Significant and exciting developments in functionalization of un‐activation Csp3‐H bonds have continuously been made over the past few decades. This review mainly summarizes recent advances on direct Csp3‐H bond functionalization for the formation of C‐C and C‐heteroatom bond under transition‐metal‐ catalysed and metal‐free conditions.
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